S fazında etkili topoizomeraz inhibitörleri

Topoisomerase inhibitors (S phase)    

I-Topoisomerase I inhibitors; Camptotheca (Belotecan, Camptothecin, Cositecan, Etirinotecan,  pegol, Exatecan, Gimatecan, Irinotecan, Lurtotecan, Rubitecan, Silatecan, Topotecan)

II-Topoisomerase II inhibitors; Podophyllum (Etoposide, Teniposide)

III-Intercalation yaparak araya giren Topoisomerase II inhibitors  

a-Anthracyclines (Aclarubicin, Amrubicin, Daunorubicin (+cytarabine), Doxorubicin, Epirubicin, Idarubicin, Pirarubicin, Valrubicin, Zorubicin)

b-Anthracenediones (Losoxantrone, Mitoxantrone, Pixantrone), Amsacrine, Bisantrene, Crisnatol, Menogaril