1-Agonists:
Peptide: Aspartocin, Carbetocin, Cargutocin, Demoxytocin, Lipo-oxytocin-1, Merotocin, Nacartocin, Oxytocin, Vasotocin (argiprestocin);
Non-peptide: CA7, LIT-001, TC OT 39, WAY-267464, WJ0679
2-Antagonists:
Peptide: Atosiban, Tocinoic acid;
Non-peptide: Barusiban, Cligosiban, Epelsiban, Erlosiban, Nolasiban, Retosiban
3-Catabolism inhibitors:
Amastatin, Bestatin (ubenimex), EDTA, L-Methionine, Leupeptin, o-Phenanthroline, Phosphoramidon, Puromycin