Kalsiyum kanal blokerleri

Voltage-gated calcium channels (VGCCs),üzerinden etki eden kalsiyum kanal blokerleri

1-L-type-selective:

Dihydropyridines:

Amlodipine

Aranidipine

Azelnidipine

Barnidipine

Clevidipine

Cronidipine

Darodipine

Dexniguldipine

Elgodipine

Elnadipine

Felodipine

Flordipine

Furnidipine

Iganidipine

Isradipine

Lacidipine

Lemildipine

Lercanidipine

Levamlodipine

Levniguldipine

Manidipine

Mepirodipine

Mesudipine

Nicardipine

Nifedipine

Niguldipine

Niludipine

Nilvadipine

Nimodipine

Nisoldipine

Nitrendipine

Olradipine

Oxodipine

Palonidipine

Pranidipine

Ryodipine (riodipine)

Sagandipine

Sornidipine

Teludipine

Tiamdipine

Trombodipine

Vatanidipine;

Diltiazem derivatives:

Clentiazem

Diltiazem

Iprotiazem

Nictiazem

Siratiazem;

Phenylalkylamines:

Anipamil

Dagapamil

Devapamil

Dexverapamil

Emopamil

Etripamil

Falipamil

Gallopamil

Levemopamil

Nexopamil

Norverapamil

Ronipamil

Tiapamil

Verapamil;

Others: AH

Brinazarone

Budiodarone

Celivarone

Cyproheptadine

Dronedarone

Fantofarone

Tetrahydropalmatine

2-N-type-selective:

ω-Conotoxins

ω-Conotoxin GVIA

Caroverine

Huwentoxin XVI

Leconotide (ω-conotoxin CVID)

Ralfinamide

Safinamide

Ziconotide (ω-conotoxin MVIIA)

3-P-type-selective:

ω-Agatoxin IVA

ω-Agatoxin IVB

4-R-type-selective: SNX-482

5-T-type-selective:

Niflumic acid

Zonisamide

6-Non-selective:

ω-Agatoxin TK

ω-Conotoxin MVIIC

Benidipine

Bepridil

Cilnidipine

Cinnarizine

Dotarizine

Efonidipine

Flunarizine

Lamotrigine

Levetiracetam

Lomerizine

Loperamide

Mibefradil

Ruthenium red

7-α2δ subunit-selective (gabapentinoids):

Methylpregabalin

Arbaclofen

Arbaclofen placarbil

Atagabalin

Baclofen

Gabapentin

Gabapentin enacarbilImagabalin

Mirogabalin

Phenibut

Pregabalin

8-4-Others/unsorted:

Bencyclane

Berbamine

Bevantolol

Canadine

Carboxyamidotriazole

Cycleanine

Dauricine

Dimeditiapramine

Diproteverine

Enpiperate

Eperisone

Elpetrigine

Ethadione

Ethanol (alcohol)

Ethosuximide

Fasudil

Fendiline

FostedilImepitoin

Lidoflazine

Magnesium

Manoalide

Mesuximide

Monatepil

Naftopidil

Ochratoxin A

Osthol

Otilonium bromide

Paramethadione

Phensuximide

Pinaverium bromide

Prenylamine

Rhynchophylline

Sesamodil

Silperisone

Sipatrigine

Terodiline

Tetrandrine

Tolperisone

Trimethadione

Valperinol